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カタログ番号 | 製品名 | 別名 | ターゲット |
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T9857 | Vasopressin | antidiuretic hormone (ADH),argipressin,arginine vasopressin (AVP) | Endogenous Metabolite |
Vasopressin (argipressin), a cyclic nine-peptide synthesized by hypothalamic neurons, is one of the hormones involved in peptide prohormone synthesis. Vasopressin is involved in the regulation process of hypothalamic-pit... | |||
T6288 | Mozavaptan | OPC31260l,OPC-31260 | Vasopressin Receptor |
Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively. | |||
T83502 | [Deamino-4-valine, 8-D-arginine]-Vasopressin | dVDAVP | |
[Deamino-4-valine, 8-D-arginine]-Vasopressin (dVDAVP) is a highly potent and specific antidiuretic agent, exhibiting prolonged effects [1] [2]. | |||
T2568 | Felypressin | Octapressin,Felypressin Acetate,PLV-2,H-[Cys-Phe-Phe-Gln-Asn-Cys]-Pro-Lys-Gly-NH2 | Vasopressin Receptor |
Felypressin (Octapressin) is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activity. | |||
T2568L | Felypressin acetate | 2-(L-Phenylalanine)-8-L-lysinevasopressin,PLV2. H-Cys-Phe-Phe-Gln-Asn-Cys-Pro-Lys-Gly-NH2 (Disulfide bond),PLV 2,PLV-2 | Vasopressin Receptor |
Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS. Felypressin acetate can be used in dental procedures. | |||
T4355 | Fuscoside | OPC 21268 | Vasopressin Receptor |
Fuscoside (OPC 21268) is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist. | |||
T7284 | Argipressin acetate (113-79-1(free base)) | Others | |
Vasopressin acetate is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values of 1.31 and 1.44 nM in A7r5 rat aortic smooth muscle... | |||
T2326 | Tolvaptan | OPC-41061 | Vasopressin Receptor , Autophagy |
Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia. | |||
T5144 | Desmopressin acetate (16679-58-6 free base) | Desmopressin acetate,DDAVP | Vasopressin Receptor |
Desmopressin acetate (16679-58-6 free base) (DDAVP) is the synthetic analog of the antidiuretic hormone arginine vasopressin. Vasopressin Receptor The antidiuretic properties of desmopressin have led to its use in polyur... | |||
TP2400 | Peptide pva | Vasopressin antisense peptide | |
Peptide pva, encoded by an RNA, is complementary to arginine vasopressin mRNA. | |||
T29178 | YM 471 | YM-471,YM471 | |
YM 471 is a non-peptide arginine vasopressin (AVP) V1A and V2 receptor antagonist with oral activity. | |||
T76573 | [8-L-arginine] deaminovasopressin | ||
[8-L-arginine] deaminovasopressin (dAVP) is a vasopressin analog [1] . | |||
T80073 | Dp[Tyr(methyl)2,Arg8]-Vasopressin | Vasopressin Receptor | |
Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1]. | |||
T40884 | SKF 100398 | d(CH2)5Tyr(Et)VAVP | |
SKF 100398, also known as d(CH2)5Tyr(Et)VAVP, is a particular analog of arginine vasopressin (AVP). It acts as a specific antagonist, specifically targeting the antidiuretic effect caused by both exogenous and endogenous... | |||
T7434 | Argipressin | Arg8-vasopressin,Vasopressin,AVP | Vasopressin Receptor |
Argipressin (Vasopressin) is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values of 1.31 and 1.44 nM in A7r5 rat aortic smooth ... | |||
T16553 | Pneumadin, rat | PNM | Others |
Pneumadin, rat (PNM) exerts a marked antidiuretic effect in animals has a functional AVP system. Pneumadin, rat (PNM) is a decapeptide, which possesses a potent stimulating effect on arginine-vasopressin (AVP) release. | |||
T83487 | [Pmp1,Tyr(OEt)2] AVP | ||
[Pmp1,Tyr(OEt)2] AVP, a linear analog of the cyclic arginine vasopressin (AVP) antagonist, retains the antagonistic properties of its parent compound while featuring modified phenylalanine (Pmp) and diethyltyrosine (Tyr(... | |||
T83501 | [Deamino-Pen1,Val4,D-Arg8]-vasopressin | Vasopressin Receptor | |
[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an antagonist of arginine-vasopressin (AVP). It effectively reduces plasma aldosterone concentration in rats and is utilized in studying the growth and steroidogenic capa... | |||
T29183 | YM-430 | YM-15430,YM-15430-1,YM-154301,YM-15430-2,YM430,YM-15430-3 | |
YM-430 is a β1 adrenergic receptor antagonist and a calcium channel antagonist. YM430 could be both an antianginal and antihypertensive agent. YM430 (10(-8)-10(-6) M) inhibited 3,4-diaminopyridine-induced rhythmic contra... | |||
T70365 | JTP-4819 | ||
JTP-4819 is a potent and selective prolyl endopeptidase (PEP) inhibitor with potential for treating Alzheimer's disease. At nanomolar concentration, JTP-4819 inhibited the degradation of substance P, arginine-vasopressin... |
カタログ番号 | 製品名 | 別名 | ターゲット |
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T21296 | Desmopressin acetate trihydrate | Desmogalen,Adiuretin,Deamino Arginine Vasopressin,Vasopressin 1-Desamino-8-arginine | |
Desmopressin acetate is a synthetic replacement for vasopressin, which reduces urine production. Medical use of Desmopressin acetate includes: (a) bed wetting; (b) diabetes insipidus; (c) nighttime urination; (d) clottin... |
カタログ番号 | 製品名 | Species | Expression System |
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TMPH-03132 | AVPR2 Protein, Pig, Recombinant (His & SUMO) | Sus scrofa (Pig) | E. coli |
Receptor for arginine vasopressin. The activity of this receptor is mediated by G proteins which activate adenylate cyclase. Involved in renal water reabsorption. AVPR2 Protein, Pig, Recombinant (His & SUMO) is expressed... |